+++
Hypothalamic and Pituitary Agents
++
Oral: 2.5-mg tablets, 5-mg capsules
++
Oral: 0.5-mg scored tablets
++
Parenteral 0.25, 3 mg/vial with diluent for subcutaneous
injection
+++
Chorionic gonadotropin (hCG) (generic,
Profasi, A.P.L., Pregnyl, others)
++
Parenteral powder to reconstitute 500, 1000, 2000 units/mL
for injection
++
Parenteral 0.1 mg for IV injection
++
++
Parenteral 0.25 mg/vial with diluent for IV or IM injection
+++
Follitropin alfa (Gonal-F)
++
Parenteral 37.5, 150 IU powder for injection
+++
Follitropin beta (FSH) (Follistim)
++
Parenteral 75 IU powder for injection
++
Parenteral 500 mcg/mL for injection
+++
Gonadorelin acetate (GnRH) (Lutrepulse)
++
Parenteral powder to reconstitute for injection via Lutrepulse
pump (0.8, 3.2 mg/vial)
+++
Gonadorelin hydrochloride (GnRH) (Factrel)
++
Parenteral 100, 500 mg for injection
++
Parenteral 3.6-, 10.8-mg subcutaneous implant
++
Parenteral 120, 300, 600 mg for subcutaneous injection
++
Parenteral 5 mg/mL for subcutaneous injection
++
Parenteral depot suspension (Lupron Depot, Depot-Ped, Depot-3,
Depot-4): lyophilized microspheres to reconstitute for IM injection
(3.75, 7.5, 11.25, 15, 22.5, 30 mg/vial)
++
Parenteral implant: 72 mg
+++
Menotropins (hMG) (Pergonal, Repronex)
++
Parenteral 75 IU FSH and 75 IU LH activity, 150 IU FSH and 150
IU LH activity, each with diluent
++
Nasal: 2 mg/mL (200 mcg/spray)
++
Parenteral 0.05, 0.1, 0.2, 0.5, 1 mg/mL for subcutaneous
or IV administration
++
Parenteral depot injection (Sandostatin LAR Depot): 10, 20, 30
mg for IM injection only
++
Oral: 0.05-, 0.25-, 1-mg tablets
+++
Protirelin (Thypinone, Relefact TRH, Thyrel
TRH)
++
Parenteral 500 mg/mL for injection
++
Parenteral 0.5, 1 mg for subcutaneous injection; 50-mcg powder
to reconstitute for intravenous injection
++
Parenteral 5, 10 mg/vial with diluent for subcutaneous
or IM injection
+++
Somatropin (Genotropin, Humatrope, Nutropin,
Nutropin Aq, Norditropin, Serostim, Saizen)
++
Parenteral 0.2, 0.4, 0.6, 0.8, 1.0, 1.2, 1.4, 1.5, 1.6, 1.8,
2, 4, 5, 5.8, 6, 8, 10, 12, 13.5, 13.8, 15, 18, 22.5, 24 mg/vial
with diluent for subcutaneous or IM injection
+++
Thyrotropin alpha (Thyrogen)
++
Parenteral 1.1 mg (4 IU)/vial with diluent for IM injection
++
Parenteral 3.75, 11.25 mg for IM injection
++
Parenteral powder to reconstitute for injection, 75, 150 IU FSH
activity per ampule
+++
Levothyroxine (T4) (generic, Levoxyl, Levo-T, Synthroid,
Unithroid)
++
Oral: 0.025-, 0.05-, 0.075-, 0.088-, 0.1-, 0.112-, 0.125-, 0.137-,
0.15-, 0.175-, 0.2-, 0.3-mg tablets
++
Parenteral 200, 500 mcg per vial (100 mcg/mL when reconstituted)
for injection
+++
Liothyronine (T3) (generic, Cytomel, Triostat)
++
Oral: 5-, 25-, 50-mcg tablets
++
+++
Liotrix (a 4:1 ratio of T4:T3)
(Thyrolar)
++
Oral: tablets containing 12.5, 25, 30, 50, 60, 100, 120, 150,
180 mcg T4 and one-fourth as much T3
+++
Thyroid desiccated (USP) (generic, Armour
Thyroid, Thyroid Strong, Thyrar, S-P-T)
++
Oral: tablets containing 15, 30, 60, 90, 120, 180, 240, 300 mg;
capsules (S-P-T) containing 120, 180, 300 mg
+++
Diatrizoate sodium (Hypaque)
++
Parenteral 25% (150 mg iodine/mL); 50% (300
mg iodine/mL) (unlabeled use)
+++
Iodide (131I) sodium (Iodotope, Sodium Iodide I131 Therapeutic)
++
Oral: available as capsules and solution
+++
Iopanoic acid (Telepaque)
++
Oral: 500-mg tablets (unlabeled use)
+++
Ipodate sodium (Oragrafin Sodium, Bilivist)
++
Oral: 500-mg capsules (unlabeled use)
++
++
Oral solution (generic, SSKI): 1 g/mL
++
Oral solution (Lugol solution): 100 mg/mL potassium
iodide plus 50 mg/mL iodine
++
Oral syrup (Pima): 325 mg/5 mL
++
Oral controlled-action tablets (Iodo-Niacin): 135 mg potassium
iodide plus 25 mg niacinamide hydroiodide
++
Oral potassium iodide tablets (generic, IOSAT, RAD-Block, Thyro-Block):
65, 130 mg
++
+++
Thyrotropin; Recombinant Human TSH (Thyrogen)
++
Parenteral 0.9 mg per vial
+++
Conjugated Estrogens (Premarin)
++
Oral: 0.3-, 0.625-, 0.9-, 1.25- 2.5-mg tablets
++
Parenteral 25 mg/5 mL for IM, IV injection
++
Vaginal: 0.625 mg/g cream base
+++
Dienestrol (Ortho Dienestrol, Dv)
++
+++
Diethylstilbestrol Diphosphate (Stilphostrol)
++
++
Parenteral 50 mg/mL injection
+++
Esterified Estrogens (Menest, Estratab)
++
Oral: 0.3-, 0.625-, 1.25-, 2.5-mg tablets
+++
Estradiol Cypionate in Oil (Generic, Depo-Estradiol
Cypionate)
++
Parenteral 5 mg/mL for IM injection
+++
Estradiol (Generic, Estrace)
++
Oral: 0.5-, 1-, 2-mg tablets
++
+++
Estradiol Transdermal (Estraderm, Others)
++
Transdermal: patches with 0.025, 0.0375, 0.05, 0.075, 0.1 mg/d
release rates
+++
Estradiol Valerate in Oil (Generic)
++
Parenteral 10, 20, 40 mg/mL for IM injection
++
Oral contraceptives are listed in Table 22–3.
+++
Estrone Aqueous Suspension (Generic, Kestrone
5)
++
Parenteral 5 mg/mL for injection
++
Oral: 0.625-, 1.25-, 2.5-, 5-mg tablets
++
Vaginal: 1.5 mg/g cream base
++
Oral: 0.02-, 0.05-, 0.5-mg tablets
++
Kit for subcutaneous implant; 1 rod of 68 mg
+++
Hydroxyprogesterone Caproate (Generic,
Hylutin)
++
Parenteral 125, 250 mg/mL for IM injection
++
Oral: 2.5-, 5-, 10-mg tablets
++
Parenteral (Depo-Provera): 150, 400 mg/mL for IM injection
+++
Megestrol Acetate (Generic, Megace)
++
Oral: 20-, 40-mg tablets; 40 mg/mL suspension
+++
Norethindrone Acetate (Generic, Aygestin)
++
+++
Norgestrel (Ovrette) (Also Table 22–3)
++
++
++
++
Parenteral 50 mg/mL in oil for IM injection
+++
Androgens and Anabolic Steroids
++
Oral: 2-, 5-, 10-mg tablets
++
Oral: 10-, 25-mg tablets; 10-mg capsules; 10-mg buccal tablets
++
Parenteral 200 mg/mL injection
+++
Nandrolone Decanoate (Deca-Durabolin,
Others)
++
Parenteral 100, 200 mg/mL in oil for injection
++
++
+++
Stanozolol (Winstrol)
++
+++
Testolactone (Teslac)
++
+++
Testosterone Aqueous (Generic, Others)
++
Parenteral 25, 50, 100 mg/mL suspension for IM
+++
Testosterone Cypionate in Oil (Generic,
Others)
++
Parenteral 100, 200 mg/mL for IM injection
+++
Testosterone Enanthate in Oil (Generic)
++
Parenteral 200 mg/mL for IM injection
+++
Testosterone Propionate in Oil (Generic,
Testex)
++
Parenteral 100 mg/mL for IM injection
++
Testosterone transdermal system
++
Patch (Testoderm): 4, 5, 6 mg/24 h release rate
++
Patch (Androderm): 2.5, 5 mg/24 h release rate
++
Gel (Androgel): 25, 50 mg total
++
Testosterone pellets (Testopel)
++
Parenteral 75 mg/pellet for parenteral injection (not
IV)
+++
SERMs, Antagonists, and Inhibitors
++
++
+++
Clomiphene (Generic, Clomid, Serophene,
Milophene)
++
+++
Danazol (Generic, Danocrine)
++
Oral: 50-, 100-, 200-mg capsules
++
++
++
Oral: 1-mg tablets (Propecia); 5-mg tablets (Proscar)
++
++
Parenteral 50 mg/mL for IM injection
++
++
++
Oral: 50-, 150-mg tablets
++
+++
Tamoxifen (Generic, Nolvadex)
++
++